muz1k schreef:Waar zou dit spulletje nuttig voor zijn? Slapen of om vooral angstgevoelens te verminderen?
Etizolam a thienodiazepine benzodiazepine derivative, is absorbed fairly rapidly with peak plasma levels achieved between 30 minutes and 2 hours and has a mean elimination half life of about 3 and a half hours. However, its pharmacologically active metabolite alpha-hydroxyetizolam which has the same potency as etizolam is eliminated more slowly with a mean half life of just over 8 hours. So it can be classified as a short-medium action benzodiazepine. Etizolam possesses potent hypnotic properties. Etizolam acts as a full agonist at the benzodiazepine receptor to produce its range of therapeutic as well as adverse effects. Similar to other benzodiazepines etizolam binds unselectively to benzodiazepine receptor subtypes.
In addition etizolam unlike most other benzodiazepines (some of which can increase levels of estradiol) has prolactogenic effects leading to an increase in prolactin blood levels.
According to the Italian P.I. sheet etizolam belongs to a new class of diazepines, thienotriazolodiazepines. This new class is easily oxidized, rapidly metabolized, and has a lower risk of accumulation, even after prolonged treatment. Etizolam has an anxiolytic action about 6 times greater than that of diazepam. Etizolam produces, especially at higher dosages, a reduction in time taken to fall asleep, an increase in total sleep time and a reduction in the number of awakenings. During tests there were not substantial changes in deep sleep. There is a reduction of REM sleep. In EEG tests of healthy volunteers Etizolam showed some characteristics of tricyclic antidepressants.
Lip schreef:In addition etizolam has prolactogenic effects leading to an increase in prolactin blood levels.
wikipedia schreef:In men, the most common symptoms of hyperprolactinaemia are decreased libido, erectile dysfunction, infertility and Gynecomastia.
PoisonDrink schreef:Lip schreef:In addition etizolam has prolactogenic effects leading to an increase in prolactin blood levels.wikipedia schreef:In men, the most common symptoms of hyperprolactinaemia are decreased libido, erectile dysfunction, infertility and Gynecomastia.
Maar zo'n vaart zal het niet lopen denk ik.. Leuk prentje ook bij die laatste.
Sublimo schreef:Ik ben er erg benieuwd naar, hopelijk binnenkort eens uittesten.
Etizolam has an anxiolytic action about 6 times greater than that of diazepam.
Einstein schreef:Het is dan ook eigenlijk etizolam, zonder R In dit soort situaties blijf ik in herhaling vallen
Hoe is het te vergelijken met temazepam? Heb beide benzo's gebruikt, maar mijn hersenen lijken compleet ongevoelig te zijn voor benzo's, ofzo.
Einstein schreef:Het is dan ook eigenlijk etizolam, zonder R
Einstein schreef:Hoe is het te vergelijken met temazepam? Heb beide benzo's gebruikt, maar mijn hersenen lijken compleet ongevoelig te zijn voor benzo's, ofzo.
You that never done nothin'
But build to destroy
You play with my world
Like it's your little toy
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